Back to Energy
SupplementModerate evidenceEnergy

L-arginine

Conditionally essential amino acid with meta-analysis support for mild blood-pressure reduction and endothelial function.

Why

L-arginine is the immediate substrate for nitric oxide synthase. Meta-analyses of RCTs report modest reductions in systolic and diastolic blood pressure at doses of 4–24 g/day. Smaller bodies of work support endothelial-function improvement (flow-mediated dilation), exercise-tolerance gains in heart failure, and erectile-function improvement (often in combination with pycnogenol).

How it works

Substrate for endothelial nitric oxide synthase (eNOS), increasing nitric oxide bioavailability and promoting vasodilation. Effect is modest in healthy adults (substrate saturated) and larger in conditions with endothelial dysfunction (diabetes, hypertension, heart failure).

Expected onset · BP effects over 4–8 weeks; endothelial-function effects over 2–4 weeks

How to take

Dosage

Blood pressure: 4–9 g/day divided. Higher doses (up to 24 g/day) used in heart failure RCTs.

Timing

Divided 2–3 times daily, away from protein meals for absorption

On the label

'L-arginine HCl' or 'L-arginine free base' with stated milligrams. Sustained-release forms have better tolerability at therapeutic doses.

Ideal for

Adults with mild hypertension, endothelial-dysfunction risk factors, or seeking endothelial-supportive nutrition. Combined preparations with citrulline or pycnogenol have additional erectile-function evidence.

Safety

Caution after acute myocardial infarction, one RCT (VINTAGE MI) reported increased mortality on L-arginine post-MI. Avoid in herpes simplex flares (arginine supports viral replication in vitro). Caution with antihypertensives, PDE5 inhibitors, and anticoagulants. GI side effects common at high doses. Pregnancy: limited data.

Evidence

At a glance

Dong 2011 Am Heart J meta-analysis (11 RCTs, n=387): oral L-arginine reduced systolic BP by 5.4 mmHg and diastolic by 2.7 mmHg vs placebo. VINTAGE MI 2006 RCT raised a specific safety signal post-MI, 8.6% mortality on L-arginine vs 0% on placebo over 6 months, leading to avoidance recommendation in that setting. Outside post-MI, effect is real but modest.

Where to get it

Shop L-arginine on Amazon

Sponsored · As an Amazon Associate, Healicus earns from qualifying purchases.